A New Formyl Peptide Receptor-1 Antagonist Conjugated Fullerene Nanoparticle for Targeted Treatment of Degenerative Disc Diseases
نویسندگان
چکیده
منابع مشابه
A novel nonpeptide ligand for formyl peptide receptor-like 1.
Formyl peptide receptor-like 1 (FPRL1) is a G protein-coupled receptor that binds natural and synthetic peptides as well as lipoxin A(4) and mediates important biological functions. To facilitate its pharmacological characterization, we screened a compound library and identified a substituted quinazolinone (Quin-C1, 4-butoxy-N-[2-(4-methoxy-phenyl)-4-oxo-1,4-dihydro-2H-quinazolin-3-yl]-benzamid...
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ژورنال
عنوان ژورنال: ACS Applied Materials & Interfaces
سال: 2019
ISSN: 1944-8244,1944-8252
DOI: 10.1021/acsami.9b11783